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Antipain

SIGMA/10791 - >50000 U/mg

Synonym: [(S)-1-Carboxy-2-phenylethyl]carbamoyl-L-arginyl-L-valyl-argininal

CAS Number: 37691-11-5
Empirical Formula (Hill Notation): C27H44N10O6
Molecular Weight: 604.70
EC Number: 253-631-0
MDL Number: MFCD00135959
Linear Formula: C27H44N10O6
Product Type: Chemical
Catalog Number PKG Qty. Price Quantity
45-10791-5MG 5 mg
 $130.00
1/EA		 Add To Favorites
45-10791-25MG 25 mg
 $486.00
1/EA		 Add To Favorites

 

InChI 1S/C27H44N10O6/c1-16(2)21(23(40)34-18(15-38)10-6-12-32-25(28)29)37-22(39)19(11-7-13-33-26(30)31)35-27(43)36-20(24(41)42)14-17-8-4-3-5-9-17/h3-5,8-9,15-16,18-21H,6-7,10-14H2,1-2H3,(H,34,40)(H,37,39)(H,41,42)(H4,28,29,32)(H4,30,31,33)(H2,35,36,43)/t18?,19-,20-,21-/m0/s1
InChI key SDNYTAYICBFYFH-KTYMLHDXSA-N
mode of action enzyme | inhibits
Quality Level 100 
SMILES string [H]C(=O)C(CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)N[C@@H](Cc1ccccc1)C(O)=O)C(C)C
specific activity >50000 U/mg
storage temp. −20°C
Biochem/physiol Actions: Inhibits serine/cysteine proteases and some trypsin-like proteases. Compare activity to that of leupeptin. Used to evaluate the role of proteases in cell transformations. Used to help identify new proteases.
Biochem/physiol Actions: Reversible inhibitor of serine/cysteine proteases and some trypsin-like serine proteases. Its action resembles leupeptin; however, its plasmin inhibition is less and its cathepsin A inhibition is more than that observed with leupeptin. Chronic administration can reduce the frequency of chemically induced transformation in BALB/c-/3T3 cells.
General description: Chemical structure: peptide
Other Notes: 1 U corresponds to the amount of inhibitor which reduces the trypsin activity by 1 BAEE-U. (1 BAEE-U is the amount of enzyme which increases the absorbance at 253 nm by 0.001 per minute at pH 7.6 and 25°C; BAEE, Cat. No. 12880, as substrate)
Other Notes: Protease inhibitor
Packaging: Bottomless glass bottle. Contents are inside inserted fused cone.
Symbol GHS07  GHS07
Signal word Warning
Hazard statements H302
RIDADR NONH for all modes of transport
WGK Germany WGK 3
Flash Point(F) Not applicable
Flash Point(C) Not applicable
activity specific activity: >50000 U/mg
Storage Temp. −20°C
UNSPSC 12352202

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