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Enalaprilat dihydrate

SIGMA/E9658 - ≥98% (HPLC)

Synonym: (2S)-1-[(2S)-2-[[(1S)-1-Carboxy-3-phenyl-propyl]amino]propanoyl]pyrrolidine-2-carboxylic acid; Vasotec

CAS Number: 84680-54-6
Empirical Formula (Hill Notation): C18H24N2O5 ·2H2O
Molecular Weight: 384.42
EC Number: 278-459-3
MDL Number: MFCD00941393
Linear Formula: C18H24N2O5 ·2H2O
Product Type: Chemical
Catalog Number PKG Qty. Price Quantity
45-E9658-5MG 5 mg
 $148.00
1/EA		 Add To Favorites
45-E9658-25MG 25 mg
 $566.00
1/EA		 Add To Favorites

 

assay ≥98% (HPLC)
InChI 1S/C18H24N2O5.2H2O/c1-12(16(21)20-11-5-8-15(20)18(24)25)19-14(17(22)23)10-9-13-6-3-2-4-7-13;;/h2-4,6-7,12,14-15,19H,5,8-11H2,1H3,(H,22,23)(H,24,25);2*1H2/t12-,14-,15-;;/m0../s1
InChI key MZYVOFLIPYDBGD-MLZQUWKJSA-N
originator Merck & Co., Inc., Kenilworth, NJ, U.S.
Quality Level 100 
SMILES string O.O.C[C@H](N[C@@H](CCc1ccccc1)C(O)=O)C(=O)N2CCC[C@H]2C(O)=O
solubility DMSO: 64 mg/mL
  H2O: 14 mg/mL at 60 °C (warming for 5 minutes)
storage temp. room temp
Biochem/physiol Actions: Enalapril, the ethyl ester of enalaprilat exhibits slight pharmacological activity until it is hydrolyzed in the liver to enalaprilat. Enalaprilat, a IV form of an angiotensin-converting-enzyme inhibitor (ACE) prevents the transformation of angiotensin I to angiotensin II, a potent vasoconstrictor.
Biochem/physiol Actions: Enalaprilat is an inhibitor of angiotensin converting enzyme (ACE), antihypertensive, and a Bradykinin B1 receptor activator.
Biochem/physiol Actions: Enalaprilat is an inhibitor of angiotensin converting enzyme (ACE), antihypertensive, and a Bradykinin B1 receptor activator. Enalaprilat has nM potency versus ACE and also activates B1 receptors to release NO.
Features and Benefits: This compound is featured on the Angiotensin Receptors  and Bradykinin Receptors  pages of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here .
Features and Benefits: This compound was developed by Merck & Co., Inc., Kenilworth, NJ, U.S. . To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here .
Packaging: 5, 25 mg in glass bottle
RIDADR NONH for all modes of transport
WGK Germany WGK 3
Flash Point(F) Not applicable
Flash Point(C) Not applicable
Purity ≥98% (HPLC)
Storage Temp. room temp
UNSPSC 12352200

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