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NIDA-41020

SIGMA/N8162 - ≥97% (HPLC), solid

Synonym: 1-(2,4-Dichlorophenyl)-5-(4-methoxyphenyl)-4-methyl-N-(1-piperidinyl)-1H-pyrazole-3-carboxamide

CAS Number: 502486-89-7
Empirical Formula (Hill Notation): C23H24Cl2N4O2
Molecular Weight: 459.37
MDL Number: MFCD08277026
Linear Formula: C23H24Cl2N4O2
Product Type: Chemical
Catalog Number PKG Qty. Price Quantity
45-N8162-50MG 50 mg
 $691.00
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assay ≥97% (HPLC)
color off-white
form solid
InChI 1S/C23H24Cl2N4O2/c1-15-21(23(30)27-28-12-4-3-5-13-28)26-29(20-11-8-17(24)14-19(20)25)22(15)16-6-9-18(31-2)10-7-16/h6-11,14H,3-5,12-13H2,1-2H3,(H,27,30)
InChI key KWDBQJRWPWTGPF-UHFFFAOYSA-N
Quality Level 100 
SMILES string COc1ccc(cc1)-c2c(C)c(nn2-c3ccc(Cl)cc3Cl)C(=O)NN4CCCCC4
solubility DMSO: ~16 mg/mL
  H2O: insoluble
storage temp. 2-8°C
Biochem/physiol Actions: NIDA-41020 is a CB1 cannabinoid receptor antagonist. NIDA-41020 is structurally similar to Rimonabant, which is currently in clinical development. NIDA-41020 is less lipophilic; developed at NIDA as a potential radioligand for CB1 receptors, Ki = 4.1 nM [in comparison AM 251, AM 281, SR 141716 (Rimonabant) have Ki of 0.6, 4.5 and 1.8 nM respectively].
Biochem/physiol Actions: NIDA-41020 is a CB1 cannabinoid receptor antagonist.
Purity ≥97% (HPLC)
Storage Temp. 2-8°C
UNSPSC 12352200

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