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MCOPPB trihydrochloride hydrate

SIGMA/PZ0159 - >98% (HPLC)

Synonym: 1-[1-(1-Methylcyclooctyl)-4-piperidinyl]-2-[(3R)-3-piperidinyl]-1H-benzimidazole trihydrochloride hydrate

CAS Number: 1028969-49-4 (free base)
Empirical Formula (Hill Notation): C26H40N4 · 3 HCl · xH2O
Molecular Weight: 518.01 (anhydrous basis)
Linear Formula: C26H40N4 · 3 HCl · xH2O
Product Type: Chemical
Catalog Number PKG Qty. Price Quantity
45-PZ0159-5MG 5 mg
 $162.00
1/EA		 Add To Favorites
45-PZ0159-25MG 25 mg
 $603.00
1/EA		 Add To Favorites

 

assay >98% (HPLC)
color white to tan
form powder
InChI 1S/C26H40N4.3ClH.H2O/c1-26(15-7-3-2-4-8-16-26)29-18-13-22(14-19-29)30-24-12-6-5-11-23(24)28-25(30)21-10-9-17-27-20-21;;;;/h5-6,11-12,21-22,27H,2-4,7-10,13-20H2,1H3;3*1H;1H2
InChI key UQBVSGBDJOJHIP-UHFFFAOYSA-N
Quality Level 100 
SMILES string O.Cl.Cl.Cl.CC1(CCCCCCC1)N2CCC(CC2)n3c(nc4ccccc34)[C@@H]5CCCNC5
solubility H2O: ≥13 mg/mL
storage condition desiccated
storage temp. room temp
Biochem/physiol Actions: MCOPPB trihydrochloride is a potent non-peptide nociceptin/orphanin FQ peptide (NOP)-receptor full agonist [or opioid-receptor-like-1 (ORL1) receptor agonist]. MCOPPB is the most potent novel non-peptide NOP full agonist in vitro and an orally potent anxiolytic in the mice. It inhibited signaling through the NOP receptor in the mouse brain, suggesting that it penetrated into the brain after it was orally administered. It did not affect locomotor activity or memory, nor did it contribute to ethanol-induced hypnosis.
Biochem/physiol Actions: Potent non-peptide nociceptin/orphanin FQ peptide (NOP)-receptor full agonist [or opioid-receptor-like-1 (ORL1) receptor agonist.
Features and Benefits: This compound is featured on the Opioid Receptors  page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here .
Packaging: 5, 25 mg in glass bottle
RIDADR NONH for all modes of transport
WGK Germany WGK 3
Flash Point(F) Not applicable
Flash Point(C) Not applicable
Purity >98% (HPLC)
Storage Temp. room temp
UNSPSC 51111800

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