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CP-101606 mesylate

SIGMA/PZ0255 - ≥98% (HPLC)

Synonym: (1S,2S)-1-(4-Hydroxy-phenyl)-2-(4-hydroxy-4-phenylpiperidino)-1-propanol mesylate; (1S,2S)-1-(4-Hydroxyphenyl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)-1-propanol mesylate; CP-101,60 mesylate; CP-101606-27; Traxoprodil mesylate

CAS Number: 188591-67-5
Empirical Formula (Hill Notation): C20H25NO3 · CH4O3S
Molecular Weight: 423.52
MDL Number: MFCD12546332
Linear Formula: C20H25NO3 · CH4O3S
Product Type: Chemical
Catalog Number PKG Qty. Price Quantity
45-PZ0255-5MG 5 mg
 $126.00
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45-PZ0255-25MG 25 mg
 $495.00
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This picture is provided solely for illustration purposes, it may have been created or edited with AI. Optical properties of the actual product may deviate. Relevant product information is printed on labeled products and other accompanying or available information material.
This image depicts PZ0255-25MG.

 

assay ≥98% (HPLC)
color white to beige
form powder
InChI 1S/C20H25NO3.CH4O3S/c1-15(19(23)16-7-9-18(22)10-8-16)21-13-11-20(24,12-14-21)17-5-3-2-4-6-17;1-5(2,3)4/h2-10,15,19,22-24H,11-14H2,1H3;1H3,(H,2,3,4)/t15-,19+;/m0./s1
InChI key OZBWUANKVIMZIA-WRRDZZDISA-N
Quality Level 100 
SMILES string OC1=CC=C([C@H](O)[C@H](C)N2CCC(O)(C3=CC=CC=C3)CC2)C=C1.CS(=O)(O)=O
solubility DMSO: 20 mg/mL, clear
storage temp. room temp
Biochem/physiol Actions: CP-101,606 is an NR2B (N-methyl D-aspartate receptor subtype 2B) subunit antagonist, that can increase dyskinesia. It reduces Ca2+/calmodulin-dependent protein kinase II level, at threonine-286 hyperphosphorylation (pCaMKII-Thr286). It has no effect on the α1-adrenergic receptors. CP-101,606 has the ability to inhibits the habits, stimulated by cocaine. It also possesses hallucinogenic properties.
Biochem/physiol Actions: CP-101606 mesylate (Traxoprodil mesylate) is a potent noncompetitive antagonist of N-methyl-D-aspartate (NMDA) receptors, selective for the NR2B subunit. CP-101606 mesylate has been shown to be neuroprotective in animal models of brain injury and stroke.
Packaging: 5, 25 mg in glass bottle
Purity ≥98% (HPLC)
Storage Temp. room temp
UNSPSC 51111800

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