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GW-803430

SIGMA/SML0230 - ≥98% (HPLC)

Synonym: 6-(4-chloro-phenyl)-3-[3-methoxy-4-(2-pyrrolidin-1-yl-ethoxy)-phenyl]-3H-thieno[3,2-d]pyrimidin-4-one; GW-3430; GW-803430A

CAS Number: 515141-51-2
Empirical Formula (Hill Notation): C25H24ClN3O3S
Molecular Weight: 481.99
Linear Formula: C25H24ClN3O3S
Product Type: Chemical
Catalog Number PKG Qty. Price Quantity
45-SML0230-5MG 5 mg
 $92.10
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assay ≥98% (HPLC)
color white to beige
form powder
InChI 1S/C25H24ClN3O3S/c1-31-22-14-19(8-9-21(22)32-13-12-28-10-2-3-11-28)29-16-27-20-15-23(33-24(20)25(29)30)17-4-6-18(26)7-5-17/h4-9,14-16H,2-3,10-13H2,1H3
InChI key MWULMTACIBZPGN-UHFFFAOYSA-N
originator GlaxoSmithKline
Quality Level 100 
SMILES string [s]1c2c(nc[n]([c]2=O)c4cc(c(cc4)OCCN5CCCC5)OC)cc1c3ccc(cc3)Cl
solubility DMSO: ≥4 mg/mL at warmed to 60 °C
storage temp. 2-8°C
Application: GW-803430 may be used in MCHR1-mediated cell signaling studies.
Biochem/physiol Actions: GW-803430 antagonizes central MCHR1 and produces anxiolytic, anti-depressant and anti-obesity effects in rats and mice. It also controls the alcohol-seeking behavior in rats and is a promising treatment for alcohol use-related disorders.
Biochem/physiol Actions: GW-803430 is a centraly active and selective melanin-concentrating hormone receptor (MCHR) 1 antagonist
Features and Benefits: This compound is featured on the Melanin-Concentrating Hormone Receptors  page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here .
Features and Benefits: This compound was developed by GlaxoSmithKline . To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here .
Packaging: 5, 25 mg in glass bottle
Purity ≥98% (HPLC)
Storage Temp. 2-8°C
UNSPSC 51111800

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