PT-S58
SIGMA/SML0410 - ≥98% (HPLC)
Synonym: 2-
CAS Number: 1356497-92-1
Empirical Formula (Hill Notation): C17H22N2O5S2
Molecular Weight: 398.50
MDL Number: MFCD22666395
Linear Formula: C17H22N2O5S2
Product Type: Chemical
assay | ≥98% (HPLC) |
color | white to beige |
form | powder |
InChI | 1S/C17H22N2O5S2/c1-17(2,3 |
InChI key | JSUWAIOZKBYWCJ-UHFFFAOYSA |
Quality Level | 100 ![]() |
SMILES string | COC1=CC(NC(C)(C)C)=CC=C1N |
solubility | DMSO: 10 mg/mL (warmed; clear solution) |
storage temp. | 2-8°C |
Biochem/physiol Actions: | PT-S58 is a PPAR β/δ full antagonist, and a derivative of GSK0660. PT-S58 has a three-fold higher affinity for the receptor than GSK0660 and is a potent inhibitor of agonist-induced target gene expression. Unlike GSK0660, PT-S58 blocks the recruitment co-repressor molecules such as SMRT. |
Features and Benefits: | This compound is featured on the Nuclear Receptors (Non-Steroids) ![]() ![]() ![]() |
Packaging: | 5, 25 mg in glass bottle |
RIDADR | NONH for all modes of transport |
WGK Germany | WGK 3 |
Flash Point(F) | Not applicable |
Flash Point(C) | Not applicable |
Purity | ≥98% (HPLC) |
Storage Temp. | 2-8°C |
UNSPSC | 12352200 |