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PT-S58

SIGMA/SML0410 - ≥98% (HPLC)

Synonym: 2-Thiophenecarboxylic acid, 3-[[[4-[(1,1-dimethylethyl)amino]-2-methoxyphenyl]amino]sulfonyl]-, methyl ester

CAS Number: 1356497-92-1
Empirical Formula (Hill Notation): C17H22N2O5S2
Molecular Weight: 398.50
MDL Number: MFCD22666395
Linear Formula: C17H22N2O5S2
Product Type: Chemical
Catalog Number PKG Qty. Price Quantity
45-SML0410-5MG 5 mg
 $163.00
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45-SML0410-25MG 25 mg
 $0.00
1/EA
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assay ≥98% (HPLC)
color white to beige
form powder
InChI 1S/C17H22N2O5S2/c1-17(2,3)18-11-6-7-12(13(10-11)23-4)19-26(21,22)14-8-9-25-15(14)16(20)24-5/h6-10,18-19H,1-5H3
InChI key JSUWAIOZKBYWCJ-UHFFFAOYSA-N
Quality Level 100 
SMILES string COC1=CC(NC(C)(C)C)=CC=C1NS(C2=C(C(OC)=O)SC=C2)(=O)=O
solubility DMSO: 10 mg/mL (warmed; clear solution)
storage temp. 2-8°C
Biochem/physiol Actions: PT-S58 is a PPAR β/δ full antagonist, and a derivative of GSK0660. PT-S58 has a three-fold higher affinity for the receptor than GSK0660 and is a potent inhibitor of agonist-induced target gene expression. Unlike GSK0660, PT-S58 blocks the recruitment co-repressor molecules such as SMRT.
Features and Benefits: This compound is featured on the Nuclear Receptors (Non-Steroids)  and Nuclear Receptors (PPARs)  pages of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here .
Packaging: 5, 25 mg in glass bottle
RIDADR NONH for all modes of transport
WGK Germany WGK 3
Flash Point(F) Not applicable
Flash Point(C) Not applicable
Purity ≥98% (HPLC)
Storage Temp. 2-8°C
UNSPSC 12352200

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