Advanced Search



ENMD-1068 hydrochloride

SIGMA/SML1039 - ≥97% (HPLC)

Synonym: 6-Amino-1-[4-(3-methyl-1-oxobutyl)-1-piperazinyl]-1-hexanone hydrochloride

CAS Number: 789488-77-3 (free base)
Empirical Formula (Hill Notation): C15H29N3O2 · HCl
Molecular Weight: 319.87
Linear Formula: C15H29N3O2 · HCl
Product Type: Chemical
Catalog Number PKG Qty. Price Quantity
45-SML1039-5MG 5 mg
 $131.00
1/EA		 Add To Favorites
45-SML1039-25MG 25 mg
 $525.00
1/EA		 Add To Favorites
This image is provided for informative purposes only and does not represent an actual product label. It should not be used as a substitute for official product labeling.

 

assay ≥97% (HPLC)
color white to beige
form powder
InChI 1S/C15H29N3O2/c1-13(2)12-15(20)18-10-8-17(9-11-18)14(19)6-4-3-5-7-16/h13H,3-12,16H2,1-2H3
InChI key VRZYMMVEALDDBH-UHFFFAOYSA-N
Quality Level 100 
SMILES string N1(CCN(CC1)C(=O)CCCCCN)C(=O)CC(C)C
solubility H2O: 25 mg/mL, clear
storage condition desiccated
storage temp. 2-8°C
Application: ENMD-1068 hydrochloride has been used as a protease-activated receptor 2 (PAR2) antagonist to determine the pathway responsible for paw edema induced by Crotalus durissus terrificus venom serine protease (Cdtsp 2).
Biochem/physiol Actions: ENMD-1068 hydrochloride exhibits anti-angiogenic and anti-inflammatory activities.
Biochem/physiol Actions: ENMD-1068 is an antagonist of protease-activated receptor 2 (PAR2).
Biochem/physiol Actions: ENMD-1068 is an antagonist of protease-activated receptor 2 (PAR2). The compound blocks TNFα production in synovial explants from patients with arthritis, and inhibits mast cell tryptase-induced recruitment of eosinophils into the pleural cavity of mice.
Packaging: 5, 25 mg in glass bottle
Symbol GHS07  GHS07
Signal word Warning
Hazard statements H302
Hazard Codes Xn
Risk Statements 22
Safety Statements 46
RIDADR NONH for all modes of transport
WGK Germany WGK 3
Flash Point(F) Not applicable
Flash Point(C) Not applicable
Purity ≥97% (HPLC)
Storage Temp. 2-8°C
UNSPSC 51111800

The following items have been added to your cart:

Choose a favorite list for this item:
Catalog Number Description Price
$

Returns/Order support

Please fill out the form below if you want to request order support from Krackeler Scientific.


Quick Order

* Required


New Year Price Updates

We are currently working diligently to update our website pricing information for the New Year. If you place an order, you will be acknowledged with any corrected pricing. If you'd like the most current information sooner, please don't hesitate to drop us an email or give us a call and we'd be happy to assist. Thank you for your patience while we are updating.

800-334-7725
office@krackeler.com


Play Video

To Request a Quote

  1. Search or Browse for items and add to them to your Shopping Cart.
  2. Click the "Request Quote" button at the bottom of the Shopping Cart page.
  3. Fill out required fields.
  4. Optionally you can convert to standard checkout mode by choosing a payment type.
  5. Click "Request Quote" at the bottom of the page.

You will be contacted with a quote.

To Order From a Quote

  1. Register and login to the website.
  2. Receive a quote from your sales representative or customer service.
  3. Have your copy of the quote in hand.
  4. Visit our quote module to search for your quote.
Back to Top