Eltoprazine hydrochloride
SIGMA/SML1526 - ≥98% (HPLC)
Synonym: 1-
CAS Number: 98206-09-8
Empirical Formula (Hill Notation): C12H16N2O2 · HCl
Molecular Weight: 256.73
MDL Number: MFCD06245586
Linear Formula: C12H16N2O2 · HCl
Product Type: Chemical
assay | ≥98% (HPLC) |
color | white to beige |
form | powder |
InChI | 1S/C12H16N2O2.ClH/c1-2-10 |
InChI key | JFSOSUNPIXJCIX-UHFFFAOYSA |
Quality Level | 100 |
SMILES string | [H]Cl.C1(OCCO2)=C2C(N3CCN |
solubility | H2O: 10 mg/mL, clear |
storage temp. | room temp |
Biochem/physiol Actions: | Eltoprazine hyrochloride is a serotonin 5-HT1A/1B receptor agonist that has been shown to reduce L-DOPA-induced dyskinesias in in experimental models of Parkinson′s Disease and in human patients. It has Ki values for 5-HT1A, 5-HT1B and 5-HT1C receptors of 40 nM and 52 nM, respectively. |
General description: | Eltoprazine, a serotonergic agent, possesses specific anti-aggressive (serenic) properties in various animal models without triggering sedation, motor disturbances, or muscle relaxation. |
Packaging: | 5, 25 mg in glass bottle |
Symbol | GHS06 |
Signal word | Danger |
Hazard statements | H301 - H315 - H319 - H335 |
Precautionary statements | P301 + P310 + P330 - P302 + P352 - P305 + P351 + P338 |
RIDADR | UN 2811 6.1 / PGIII |
WGK Germany | WGK 3 |
Flash Point(F) | Not applicable |
Flash Point(C) | Not applicable |
Purity | ≥98% (HPLC) |
Storage Temp. | room temp |
UNSPSC | 12352200 |