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Tianeptine sodium salt hydrate

SIGMA/T1692 - ≥98% (HPLC), powder

Synonym: 7-[(3-Chloro-6,11-dihydro-6-methyl-dibenzo[c,f][1,2]thiazepine-11-yl)amino]heptanoic acid S,S dioxide sodium salt hydrate

CAS Number: 30123-17-2 (anhydrous)
Empirical Formula (Hill Notation): C21H24ClN2NaO4S · xH2O
Molecular Weight: 458.93 (anhydrous basis)
Linear Formula: C21H24ClN2NaO4S · xH2O
Product Type: Chemical
Catalog Number PKG Qty. Price Quantity
45-T1692-5MG 5 mg
 $346.00
1/EA		 Add To Favorites
45-T1692-25MG 25 mg
 $1250.00
1/EA		 Add To Favorites

 

assay ≥98% (HPLC)
color white to tan
form powder
InChI 1S/C21H25ClN2O4S.Na.H2O/c1-24-18-9-6-5-8-16(18)21(23-13-7-3-2-4-10-20(25)26)17-12-11-15(22)14-19(17)29(24,27)28;;/h5-6,8-9,11-12,14,21,23H,2-4,7,10,13H2,1H3,(H,25,26);;1H2/q;+1;/p-1
InChI key HNTRDGDHBBFLPG-UHFFFAOYSA-M
originator Servier
Quality Level 100 
SMILES string O.[Na+].CN1c2ccccc2C(NCCCCCCC([O-])=O)c3ccc(Cl)cc3S1(=O)=O
solubility DMSO: ≥20 mg/mL
storage condition desiccated
storage temp. room temp
Application: Tianeptine sodium salt hydrate has been used as a selective serotonin reuptake enhancer (SSRE) positive control during serotonin transporter (SERT) assay in human embryonic kidney 293 cell lines.
Biochem/physiol Actions: Tianeptine is a tricyclic antidepressant that enhances serotonin uptake. This drug can affect neuroprotection, neuronal excitability, memory and anxiety. However, tianeptine is not linked to adverse psychomotor, cognitive, cardiovascular, sleep and bodyweight effects. The drug has a low tendency for abuse and has a positive pharmacokinetic profile.
Biochem/physiol Actions: Tianeptine is least involved in drug interaction as it is not metabolized by cytochrome P450 system in the liver. In hippocampus and amygdala, tianeptine is involved in glutamatergic transmission processes and elicits neuroplasticity.
Features and Benefits: This compound was developed by Servier . To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here .
General description: Tianeptine is a μ-opioid receptor (MOR) as well as a δ-opioid receptor (DOR) agonist.
Packaging: 5, 25 mg in glass bottle
Preparation Note: Tianeptine sodium salt hydrate is soluble in DMSO at a concentration that is greater than or equal to 20 mg/ml.
RIDADR NONH for all modes of transport
WGK Germany WGK 3
Flash Point(F) Not applicable
Flash Point(C) Not applicable
Purity ≥98% (HPLC)
Storage Temp. room temp
UNSPSC 12352200

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